Silver-catalyzed synthesis of 4-substituted benzofurans via a cascade oxidative coupling-annulation protocol.
نویسندگان
چکیده
A facile synthesis of 4-indole benzofurans from the one-pot reaction of 4-alkyl-2-ynylphenols and indoles via a hypervalent iodine-induced oxidative dearomatization, a silver-catalyzed cascade Michael addition-annulation, and an aromatization is reported.
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ورودعنوان ژورنال:
- Chemical communications
دوره 47 19 شماره
صفحات -
تاریخ انتشار 2011